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Issue 12, 2016
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Silver(I)-promoted C5–H phosphonation of 8-aminoquinoline amides with H-phosphonates

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Abstract

A simple and efficient protocol for silver(I)-promoted phosphonation of 8-aminoquinoline amides with dialkyl H-phosphonates has been developed, affording the desired products in moderate yields. This method features C5–H regioselectivity of 8-aminoquinoline amides, a broad substrate scope and general functional group compatibility.

Graphical abstract: Silver(i)-promoted C5–H phosphonation of 8-aminoquinoline amides with H-phosphonates

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Publication details

The article was received on 21 Jul 2016, accepted on 15 Sep 2016 and first published on 19 Sep 2016


Article type: Research Article
DOI: 10.1039/C6QO00379F
Citation: Org. Chem. Front., 2016,3, 1646-1650
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    Silver(I)-promoted C5–H phosphonation of 8-aminoquinoline amides with H-phosphonates

    M. Sun, S. Sun, H. Qiao, F. Yang, Y. Zhu, J. Kang, Y. Wu and Y. Wu, Org. Chem. Front., 2016, 3, 1646
    DOI: 10.1039/C6QO00379F

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