A new type of galactose mimetics has been synthesized following a straightforward synthetic approach based on cyclohexene olefin aziridination reactions directed by hydroxyl substituents. These enantiomerically pure galacto-configured N-aminoaziridines are potent irreversible inhibitors of Aspergillus oryzae and Escherichia coli β-galactosidases.
A. Alcaide, A. Trapero, Y. Pérez and A. Llebaria, Org. Biomol. Chem., 2015, 13, 5690 DOI: 10.1039/C5OB00532A
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