Issue 6, 2002
From the journal:

Journal of the Chemical Society, Perkin Transactions 1

Efficient regioselective synthesis of triheterocyclic compounds: imidazo[2,1-b]benzothiazoles, pyrimido[2,1-b]benzothiazolones and pyrimido[2,1-b]benzothiazoles

Cyrille Landreau,a   David Deniaud,*a   Michel Evain,b   Alain Reliqueta  and  Jean-Claude Meslina  

* Corresponding authors

a Laboratoire de Synthèse Organique, Faculté des Sciences et des Techniques, UMR C.N.R.S. 6513, BP 92208, 2, rue de la Houssinière, F44322 Nantes Cedex 03, France

b Institut des Matériaux Jean Rouxel, Laboratoire de Chimie des Solides, Faculté des Sciences et des Techniques, 2, rue de la Houssinière, BP 32 229, F-44322 Nantes Cedex 03, France

Abstract

The preparation and characterisation of triheterocyclic compounds, via annulation reactions, are described. Amidines 1 reacted with substituted bromomethyl compounds, acid chlorides, and acrylic dienophiles to afford the corresponding imidazo[2,1-b]benzothiazoles 2 and pyrimido[2,1-b]benzothiazoles 3 or 4.

Graphical abstract: Efficient regioselective synthesis of triheterocyclic compounds: imidazo[2,1-b]benzothiazoles, pyrimido[2,1-b]benzothiazolones and pyrimido[2,1-b]benzothiazoles

About
Cited by
Related
Download options Please wait...

Supplementary files

Article information

DOI
https://doi.org/10.1039/B111639H
Article type
Paper
Submitted
21 Dec 2001
Accepted
05 Feb 2002
First published
22 Feb 2002

J. Chem. Soc., Perkin Trans. 1, 2002, 741-745

Permissions

Request permissions

Efficient regioselective synthesis of triheterocyclic compounds: imidazo[2,1-b]benzothiazoles, pyrimido[2,1-b]benzothiazolones and pyrimido[2,1-b]benzothiazoles

C. Landreau, D. Deniaud, M. Evain, A. Reliquet and J. Meslin, J. Chem. Soc., Perkin Trans. 1, 2002, 741 DOI: 10.1039/B111639H

To request permission to reproduce material from this article, please go to the Copyright Clearance Center request page.

If you are an author contributing to an RSC publication, you do not need to request permission provided correct acknowledgement is given.

If you are the author of this article, you do not need to request permission to reproduce figures and diagrams provided correct acknowledgement is given. If you want to reproduce the whole article in a third-party publication (excluding your thesis/dissertation for which permission is not required) please go to the Copyright Clearance Center request page.

Read more about how to correctly acknowledge RSC content.

Spotlight

Advertisements