Issue 38, 2014

AcOH-mediated dichloroimination of indoles using chloramine-B: a facile access to 2,3-functionalized indolines

Abstract

A new and mild method for the efficient synthesis of 3,3-dichloro-2-sulfonyliminoindolines via AcOH-mediated dichloroimination of indoles using chloramine-B is presented. Application of this method to the efficient construction of pyrrolidinoindoles and N–C3 linked pyrrolidinoindolines is demonstrated.

Graphical abstract: AcOH-mediated dichloroimination of indoles using chloramine-B: a facile access to 2,3-functionalized indolines

Supplementary files

Article information

Article type
Communication
Submitted
06 Jun 2014
Accepted
12 Aug 2014
First published
13 Aug 2014

Org. Biomol. Chem., 2014,12, 7494-7497

Author version available

AcOH-mediated dichloroimination of indoles using chloramine-B: a facile access to 2,3-functionalized indolines

X. Liu, Q. Hu, Z. Yuan and P. Liu, Org. Biomol. Chem., 2014, 12, 7494 DOI: 10.1039/C4OB01179A

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