Issue 18, 2012
From the journal:

Organic & Biomolecular Chemistry

Synthesis of carbazolones and 3-acetylindoles via oxidative C–N bond formation through PIFA-mediated annulation of 2-aryl enaminones†

Xu Ban,a   Yan Pan,a   Yingfu Lin,a   Songqing Wang,*a   Yunfei Du*a  and  Kang Zhaoa  

* Corresponding authors

a Tianjin Key Laboratory for Modern Drug Deliver & High-Efficiency, School of Pharmaceutical Science and Technology, Tianjin University, Tianjin, P. R. China
E-mail: duyunfeier@tju.edu.cn, wangsq57@sina.com
Fax: +86-22-27404031
Tel: +86-22-27404031

Abstract

A series of carbazolone derivatives and 3-acetylindoles have been achieved via PIFA-mediated intramolecular cyclization of 2-aryl enaminones. This process allows the N-moiety on the side-chain to be annulated to the benzene ring via the metal-free oxidative aromatic C–N bond formation.

Graphical abstract: Synthesis of carbazolones and 3-acetylindoles via oxidative C–N bond formation through PIFA-mediated annulation of 2-aryl enaminones

About
Cited by
Related
Download options Please wait...

Supplementary files

Article information

DOI
https://doi.org/10.1039/C2OB25348H
Article type
Communication
Submitted
18 Feb 2012
Accepted
15 Mar 2012
First published
15 Mar 2012

Org. Biomol. Chem., 2012,10, 3606-3609

Permissions

Request permissions

Synthesis of carbazolones and 3-acetylindoles via oxidative C–N bond formation through PIFA-mediated annulation of 2-aryl enaminones

X. Ban, Y. Pan, Y. Lin, S. Wang, Y. Du and K. Zhao, Org. Biomol. Chem., 2012, 10, 3606 DOI: 10.1039/C2OB25348H

To request permission to reproduce material from this article, please go to the Copyright Clearance Center request page.

If you are an author contributing to an RSC publication, you do not need to request permission provided correct acknowledgement is given.

If you are the author of this article, you do not need to request permission to reproduce figures and diagrams provided correct acknowledgement is given. If you want to reproduce the whole article in a third-party publication (excluding your thesis/dissertation for which permission is not required) please go to the Copyright Clearance Center request page.

Read more about how to correctly acknowledge RSC content.

Social activity

Spotlight

Advertisements