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Issue 13, 2011
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Catalytic enantioselective synthesis of A-86929, a dopamine D1 agonist

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Abstract

A-86929, a dopamine D1 agonist was synthesized with 95% ee in five steps with overall yield of 56% viacatalytic enantioselective one-pot aziridination followed by Friedel–Crafts cyclization and a mild Pictet–Spengler cyclization protocol.

Graphical abstract: Catalytic enantioselective synthesis of A-86929, a dopamine D1 agonist

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Publication details

The article was received on 14 Jan 2011, accepted on 25 Jan 2011 and first published on 14 Feb 2011


Article type: Communication
DOI: 10.1039/C1CC10263J
Citation: Chem. Commun., 2011,47, 3981-3982
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    Catalytic enantioselective synthesis of A-86929, a dopamine D1 agonist

    S. Hajra and S. Bar, Chem. Commun., 2011, 47, 3981
    DOI: 10.1039/C1CC10263J

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