without changing your settings we'll assume you are happy to receive all RSC cookies.
You can change your cookie settings by navigating to our Privacy and Cookies page and following the instructions. These instructions
are also obtainable from the privacy link at the bottom of any RSC page.
Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zu Chong Zhi Road, Zhangjiang Hi-Tech Park, Shanghai 201203, PR China
; Fax: (+) 86 21 50807288
; Tel: (+) 86 21 50807288
Org. Biomol. Chem., 2012,10, 8953-8955
07 Sep 2012,
05 Oct 2012
First published online
09 Oct 2012
Direct C-2 amidation of indoles was reported using sulfonyl azides as the amino source to release N2 as the single byproduct. This reaction exhibits high functional group tolerance and regioselectivity, providing a variety of 2-amino substituted indoles in high to excellent yield. The procedure is robust, reliable, and compatible with water and air.
Fetching data from CrossRef. This may take some time to load.
Organic & Biomolecular Chemistry
- Information Point