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Issue 1, 2011
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The traceless Staudinger ligation for indirect 18F-radiolabelling

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Abstract

The Staudinger ligation of phosphine-substituted thioesters with 18F-fluoroethylazide has been successfully applied to access 18F-labelled molecules in radiochemical yields superior to 95%; the first fluorous variant of a Staudinger radio-ligation has been validated.

Graphical abstract: The traceless Staudinger ligation for indirect 18F-radiolabelling

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Publication details

The article was received on 10 Aug 2010, accepted on 06 Oct 2010 and first published on 22 Nov 2010


Article type: Paper
DOI: 10.1039/C0OB00564A
Citation: Org. Biomol. Chem., 2011,9, 136-140
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    The traceless Staudinger ligation for indirect 18F-radiolabelling

    L. Carroll, S. Boldon, R. Bejot, J. E. Moore, J. Declerck and V. Gouverneur, Org. Biomol. Chem., 2011, 9, 136
    DOI: 10.1039/C0OB00564A

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