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Issue 1, 2010
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Facile P,N-heterocycle synthesis via tandem aminomethylation–cyclization of H-phosphinate building blocks

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Abstract

Various heterocycles containing phosphorus and nitrogen are easily synthesized from readily available H-phosphinate building blocks. Aminomethylation of these H-phosphinates is followed by in situ cyclization through substitution or cross-coupling to produce novel heterocycles in moderate to good yields.

Graphical abstract: Facile P,N-heterocycle synthesis via tandem aminomethylation–cyclization of H-phosphinate building blocks

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Publication details

The article was received on 24 Aug 2009, accepted on 25 Sep 2009 and first published on 05 Nov 2009


Article type: Paper
DOI: 10.1039/B917428A
Citation: Org. Biomol. Chem., 2010,8, 267-273
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    Facile P,N-heterocycle synthesis via tandem aminomethylation–cyclization of H-phosphinate building blocks

    C. Queffélec and J. Montchamp, Org. Biomol. Chem., 2010, 8, 267
    DOI: 10.1039/B917428A

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