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Issue 5, 2009
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Direct C–H borylation and C–H arylation of pyrrolo[2,3-d]pyrimidines: synthesis of 6,8-disubstituted 7-deazapurines

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Abstract

Novel direct C–H borylations of 7-deazapurines to position 8 by B2pin2 under Ir catalysis were followed by Suzuki cross-couplings with aryl halides and other functional group transformations to give diverse 8-substituted 7-deazaadenines.

Graphical abstract: Direct C–H borylation and C–H arylation of pyrrolo[2,3-d]pyrimidines: synthesis of 6,8-disubstituted 7-deazapurines

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Publication details

The article was received on 06 Jan 2009, accepted on 06 Jan 2009 and first published on 14 Jan 2009


Article type: Communication
DOI: 10.1039/B900218A
Citation: Org. Biomol. Chem., 2009,7, 866-868
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    Direct C–H borylation and C–H arylation of pyrrolo[2,3-d]pyrimidines: synthesis of 6,8-disubstituted 7-deazapurines

    M. Klečka, R. Pohl, B. Klepetářová and M. Hocek, Org. Biomol. Chem., 2009, 7, 866
    DOI: 10.1039/B900218A

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